enzalutamide en · NOUN
Etymology
Etymology tree Arabic لُبَان (lubān) Proto-Indo-European *yew- Proto-Indo-European *-os Proto-Indo-European *yéwos Proto-Indo-Iranian *yáwas Sanskrit यव (yava)bor.? Proto-Austronesian *zawa Proto-Malayo-Polynesian *zawader.? Old Javanese jawa Old Javanese -i Old Javanese Jawi Javanese ꦗꦮꦶ (jawi)der. Arabic جَاوَة (jāwa) Proto-Afroasiatic Proto-Semitic Arabic ـِيّ (-iyy) Arabic جَاوِيّ (jāwiyy) Arabic لُبَان جَاوِيّ (lubān jāwiyy)bor. Catalan benjuíder. Middle French benjoinder. English benzoin English benzo- English benz- Egyptian jmnbor. Ancient Greek Ᾰ̓́μμων (Ắmmōn)bor. Latin Ammōn Latin ammoniacusder. English ammonia Proto-Indo-European *dʰeh₁-der. Proto-Italic *-iðos Latin -idusder. English -ide English amide English benzamide Proto-Indo-European *bʰel-der. Proto-Indo-European *bʰlewH-der. Proto-Indo-European *bʰluH-yé-ti? Latin fluō Proto-Indo-European *-os Proto-Indo-European *-s Proto-Indo-European *-ōs Proto-Italic *-ōs Latin -or Latin fluor Ancient Greek -ο- (-o-)der. Latin -o-bor. English -o- English fluoro- Ancient Greek ῐ̓́σος (ĭ́sos)lbor. English iso- English butyric ▲ English amide blend English butyramide English isobutyramide blend English flutamide English -lutamide English enzalutamide From (b)enza(mide) + -lutamide (“nonsteroid antiandrogen”).
Meanings
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(uncountable) A synthetic, non-steroidal pure antiandrogen developed for the treatment of metastatic castration-resistant prostate cancer.
Abiraterone and enzalutamide are newly approved drugs for CRPC patients; although, patients will still eventually relapse and the overall survival is prolonged only ~4–5 months after treatment with the AR signaling becoming active in most of these relapsed tumors.
2015 July 16, “Poly (A) Binding Protein Cytoplasmic 1 Is a Novel Co-Regulator of the Androgen Receptor”, in PLOS ONE, →DOI: